葛广波-药物代谢产物的鉴定、分析与制备.pdf

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大连化学物理研究所药用资源开发组

药物代谢产物的鉴定、分析与制备 Identification, detection and preparation of drug metabolites in eADME studies 葛广波 Lab of Pharmaceutical Resource Discovery Dalian Institute of Chemical Physics, the Chinese Academy of Sciences www.pharm.dicp.ac.cn Sep 28th, 2009

大连化学物理研究所药用资源开发组 Outline Background & research significance; Identification of drug and its metabolites; Quantification of drug and its metabolites; Methods for preparation of drug metabolites; Summary & perspectives 大连化学物理研究所药用资源开发组 Research Background Discovery Development Discovery Development Preclinical Clinical trials FDA

Target HTS Hit Lead Candidate testing ( I, II, III) approval Improvement of efficacy and safety 动物模型选择及整体PK研究 combined with ADME optimization PK参数种间放大、推导及验证 (Screening of Drug specific properties) (生

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